Contents

1. Molecular Recognition in Ligand–Protein Binding, T. Liljefors 2. Biostructure-Based Drug Design, F. S. Jørgensen and J. S. Kastrup 3. Ligand-Based Drug Design, I. Pettersson, T. Balle, and T. Liljefors 4. Chemical Biology, K. Strømgaard 5.Stereochemistry in Drug Design, M. B. Mayo-Martin and D. E. Jane 6. Natural Products in Drug Discovery, G. T. Carter 7. Imaging in Drug Discovery and Development, M. Rudin and T. Mueggler 8. Peptides and Peptidomimetics, M. Cai, V. V. Kulkarni, and V. J. Hruby 9. Prodrugs: Design and Development, A. Buur and N. Mørk 10. Metals in Medicine: Inorganic Medicinal Chemistry, H. R. Hansen and O. Farver 11. Enzyme Inhibitors: Biostructure-Based and Mechanism- Based Designs, R. A. Copeland, R. R. Gontarek, and L. Luo 12. Receptors: Structure, Function, and Pharmacology, H. Bräuner-Osborne 13. Ion Channels: Structure and Function, S.-P. Olesen and D. B. Timmermann 14. Neurotransmitter Transporters: Structure and Function, C. J. Loland and U. Gether 15. GABA and Glutamic Acid Receptor Ligands, B. Frølund and U. Madsen 16. Acetylcholine, A. A. Jensen and P. Krogsgaard-Larsen 17. Histamine Receptors, I. de Esch, H. Timmerman, and R. Leurs 18. Dopamine and Serotonin, B. Bang- Andersen and K. P. Bøgesø 19. Opioid and Cannabinoid Receptors, R. P. Clausen and H. S. Hansen 20. Hypnotics, B. Ebert and K. A. Wafford 21. Neglected Diseases, S. B. Christensen 22. Immunomodulating Agents, U. G. Sidelmann 23. Anticancer Agents, F. Björkling and L. H. Jensen 24. Antiviral Drugs, E. De Clercq 25. Antibiotics, P. Herdewijn